Type of drug | Antidopaminergic mechanism | Examples |
First-generation antipsychotics | D2R antagonism (high potency) | - Droperidol
- Flupenthixol
- Fluphenazine
- Haloperidol
- Loxapine
- Perphenazine
- Pimozide
- Thiopropazate
- Thioproperazine
- Thiothixene
- Trifluoperazine
|
D2R antagonism (low potency) | - Chlorpromazine
- Chlorprothixene
- Levomepromazine
- Mepazine
- Mesoridazine
- Methoxypromazine
- Pericyazine
- Pimozide
- Promazine
- Thioridazine
|
Second-generation antipsychotics | D2R antagonism | - Asenapine
- Clozapine*
- Iloperidone
- Lurasidone
- Olanzapine
- Paliperidone
- Quetiapine*
- Risperidone
- Sulpiride/L-sulpiride
- Ziprasidone
|
Partial D2R agonism | - Aripiprazole
- Brexpiprazole
|
Antiemetic/promotility agents | D2R antagonism | - Clebopride
- Metoclopramide
- Prochlorperazine
- Promethazine*
|
Calcium channel blockers | D2R antagonism | |
Dopamine-depleting agents | Presynaptic dopamine depletion (no DR activity) | - Deutetrabenazine
- Reserpine
- Tetrabenazine
- Valbenazine
|